Title Synthesis and HDAC inhibitory activity of pyrimidine-based hydroxamic acids /
Authors Jakubkienė, Virginija ; Valiulis, Gabrielius Ernis ; Žvirblis, Mantas ; Žvinys, Gediminas ; Zubrienė, Asta ; Matulis, Daumantas
DOI 10.15388/CCT.2019
ISBN 9786090701676
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Is Part of Chemistry and chemical technology: Lithuanian chemists conference, 2019 May 16, Lithuanian Academy of Sciences, Vilnius: conference book.. Vilnius : Vilniaus universiteto leidykla, 2019. p. 63.. ISBN 9786090701676
Keywords [eng] pyrimidines ; hydroxamic acids ; HDAC8 inhibitory activity
Abstract [eng] In continuation of our interest in the synthesis of biologically active heterocycles, a series of pyrimidine-based hydroxamic acids was prepared and evaluated as inhibitors of HDAC8.
Published Vilnius : Vilniaus universiteto leidykla, 2019
Type Conference paper
Language English
Publication date 2019